VIDRAFT AETHER-PharmaOS structure-based ensemble (gradient-boosted trees + tabular foundation model) for PKIS2 LOK and SLK kinase percent-inhibition multitask regression.
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| Test set | Target label | Metric | Score |
|---|---|---|---|
| test | LOK | r2 | 0.3660848124163182 |
| test | LOK | pearsonr | 0.6098342864597929 |
| test | LOK | spearmanr | 0.6198736514375567 |
| test | LOK | explained_var | 0.36846225246591713 |
| test | LOK | mean_squared_error | 865.7563415439454 |
| test | LOK | mean_absolute_error | 20.93428936528437 |
| test | SLK | r2 | 0.206258882170412 |
| test | SLK | pearsonr | 0.4662133766151287 |
| test | SLK | spearmanr | 0.40560215203741906 |
| test | SLK | explained_var | 0.20645265028524473 |
| test | SLK | mean_squared_error | 708.6162514281158 |
| test | SLK | mean_absolute_error | 20.406437015172205 |